The Salts Prepared from Aminopyridinium Derivatives and Saccharin as Efficient Recyclable Acylation

来源 :第九届IUPAC化学生物学国际研讨会暨第八届世界华人药物化学研讨会 | 被引量 : 0次 | 上传用户:baby3911
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  Esterification reaction is one of the most important organic reactions in the pharmaceutical industry.Homogeneous catalysis is a powerful tool in highly active and stereoselective organic transformations.It has been reported that 4-(N,N-dimethylamino)pyridine(DMAP) is an effective homogeneous catalyst for the esterification of alcohols with acid anhydrides,the ring-opening polymerization,the silylation of alcohols and others.In order to avoid spreading these harmful chemicals to the surroundings,it is important to find a recoverable catalyst that could be easily separated from the product mixture after reaction.
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