A general route towards delivering poorly soluble organometallic drugs

来源 :International Conference on Nanoscience & Technology,China 2 | 被引量 : 0次 | 上传用户:Thunder_
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  Organometallic drugs have often occupied a difficult niche in terms of therapeutic value.Bioactive metal containing compounds can demonstrate high efficacy but can also suffer from a low bioavailability.Predominantly this is as a result of poor solubility under physiological conditions which means that it is difficult to reach beneficial drug concentrations in-vivo without the dose becoming toxic and many potential antibacterial and anticancer drugs have been abandoned due to related insurmountable formulation issues.
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