【摘 要】
:
β-Enaminones and β-enamino esters,which combine the nucleophilic enamine and the electrophilic enone(ester)moieties into one molecule,represent important
【机 构】
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College of Chemistry & Chemical Engineering,Yangzhou University Yangzhou 225002
【出 处】
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中国化学会全国第十二届有机合成化学学术研讨会
论文部分内容阅读
β-Enaminones and β-enamino esters,which combine the nucleophilic enamine and the electrophilic enone(ester)moieties into one molecule,represent important synthetic building blocks and have been extensively employed as synthons for the synthesis of a wide variety of heterocycles.3-Arylamino-1-methyl-1H-pyrrole-2,5-diones,which can be easily prepared from the reaction of arylamine,dimethyl acetylenedicarboxylate and methylamine,maintain the structural character of β-enaminones and β-enamino esters.
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