【摘 要】
：
2,3-Dihydrofurans are important functionalized building blocks of natural and unnatural products because of their various biological activities,[1] sush as
【机 构】
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College of Chemistry and Molecular Engineering,Zhengzhou University,Zhengzhou,Henan 450052,China
【出 处】
：
中国化学会全国第十二届有机合成化学学术研讨会
论文部分内容阅读
2,3-Dihydrofurans are important functionalized building blocks of natural and unnatural products because of their various biological activities,[1] sush as aflatoxin B1 and clerodin.[2]Thus,the synthesis of this kind of compounds has been long-standing challenge in organic chemistry,and considerable effort has been devoted to developing efficient and selective synthetic methods to access substituted 2,3-Dihydrofurans.[3] Herein,we report a ordinary and efficient method through the Michael/Hemiketalization reaction of β,γ-Unsaturated Ketoesters and α-Hydroxyacetophenone for the synthesis of substituted 2,3-Dihydrofurans.
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