An efficient one-pot,three-component synthesis of 1,5-benzodiazepine derivatives using Ce(OTf)3-SiO2

来源 :中国化学会全国第十二届有机合成化学学术研讨会 | 被引量 : 0次 | 上传用户：xxk2010

【摘要】

：

　　1,5-Benzodiazepines are very important compounds,widely used in the last decades as anticonvulsant,antianxiety and hypnotic agents[1].The synthesis of these

【作者】

：

Liuqiannan;Wanglanzhi;

【机构】

：

The College of Chemistry and Material Science,Hebei Normal University,Shijiazhuang 050024

【出处】

：

中国化学会全国第十二届有机合成化学学术研讨会

【发表日期】

：

2015年期

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　　1,5-Benzodiazepines are very important compounds,widely used in the last decades as anticonvulsant,antianxiety and hypnotic agents[1].The synthesis of these compounds has been receiving a great deal of attention,especially its antimicrobial activity.As we known,conventional Lewis acids are very effective catalysts for a wide variety of organic reactions,but they have some disadvantages.

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An efficient one-pot,three-component synthesis of 1,5-benzodiazepine derivatives using Ce(OTf)3-SiO2

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