【摘 要】
：
An efficient synthetic method has been developed to construct benzo[b]naphtho[2,1-d]thiophene (2) via Au-catalyzed cyclizayion reaction.Treatment of 2-[2-(2-alkynylphenyl)ethynyl]thioanisole (1) under
【机 构】
：
Department of Chemistry,National Sun Yat-sen University,70 Lienhai Rd.,Kaohsiung 80424
【出 处】
：
The 24th International Society of Heterocyclic Chemistry Con
论文部分内容阅读
An efficient synthetic method has been developed to construct benzo[b]naphtho[2,1-d]thiophene (2) via Au-catalyzed cyclizayion reaction.Treatment of 2-[2-(2-alkynylphenyl)ethynyl]thioanisole (1) under 2 equivalents of NIS and 5 mol％ of Ph3PAuCl/AgSbF6 at refluxing CH2Cl2 gave compound 2 in good to excellent yields.
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