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组蛋白去乙酰化酶抑制剂(Histone deacetylases inhibitors,HDACis)是一类能够诱导细胞凋亡,抑制肿瘤生长的活性分子。目前已有三个HDACis被美国FDA批准用于治疗淋巴癌以及多发性骨髓瘤[1]。
Santacruzamate A类似物的抗肿瘤活性研究
【摘 要】
：
组蛋白去乙酰化酶抑制剂(Histone deacetylases inhibitors,HDACis)是一类能够诱导细胞凋亡,抑制肿瘤生长的活性分子。目前已有三个HDACis被美国FDA批准用于治疗淋巴癌以及多发性骨髓瘤[1]。
【机 构】
：
中山大学肿瘤防治中心/华南肿瘤学国家重点实验室,中国广州,510060
【出 处】
：
2015年全国药物化学学术会议暨第五届中英药物化学学术会议
【发表日期】
：
2015年3期
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