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【通用名】valsartan,缬沙坦【化学名】(S)N戊酰基N[[2’(1H四唑5)二苯4]甲基]缬氨酸【药理作用】在大鼠血管平滑肌细胞和人子宫肌层膜分别表达AT1和AT2受体亚型,代文竞争结合[125I]血管紧张素Ⅱ结合部位的k...
【Common name】 valsartan, valsartan 【Chemical Name】 (S) N valeryl N [2 (1H tetrazole 5 ) diphenyl 4 ] methyl] valine [Pharmacological effects] AT1 and AT2 receptor subtypes are expressed in rat vascular smooth muscle cells and human myometrial muscle membranes, respectively, and do not compete with [125I] angiotensin II binding site.