Endogenous histamine inhibits the development of morphine-induced conditioned place preference

来源 :Acta Pharmacologica Sinica | 被引量 : 0次 | 上传用户:bazzi89
下载到本地 , 更方便阅读
声明 : 本文档内容版权归属内容提供方 , 如果您对本文有版权争议 , 可与客服联系进行内容授权或下架
论文部分内容阅读
Aim:The conditioned place preference(CPP)paradigm was used to investigatethe effects of endogenous histamine on the processes leading to morphine-induced reward-seeking behavior in Sprague-Dawley rats.Methods:The modelof CPP was used to assess the rewarding effect of morphine.The levels of histamine,glutamate,γ-aminobutyric acid(GABA),dopamine(DA)and 3,4-dihydroxyphenyl-acetic acid(DOPAC)in rat brains were measured with high-performance liquidchromatography.Immunohistochemistry technique was used to observe themorphological changes of neurons.Results:Intraperitoneal injection of mor-phine(2,5 or 10 mg/kg)induced the development of CPP in a dose-dependentmanner.In addition,morphine administrations(10 mg/kg)decreased the hista-mine content and reduced the number and size of histaminergic neurons in thetuberomammillary nucleus(TM),as well as markedly increasing the DOPAC/DAratios in the ventral tegmental area(VTA)and nucleus accumbens(NAc).Intra-peritoneal injection of histidine(50,100 or 200 mg/kg)dose-dependently inhibitedthe development of morphine-induced CPP.Bilateral lesions of the TM,whichdecreased the histamine levels in the VTA and NAc,potentiated the developmentof CPP induced by morphine(1 mg/kg,a dose that produced no appreciable effectwhen given alone)and increased the DOPAC/DA ratios in the VTA and NAc,butdid not change the glutamate or GABA levels in these nuclei.Histidine reversedthe effects of the TM lesions.Conclusion:These results indicate that endog-enous histamine plays a role in inhibiting the development of morphine-inducedreward-seeking behavior,and the inhibition may involve the modulation of dopa-minergic activity. Aim: The conditioned place preference (CPP) paradigm was used to investigate the effects of endogenous histamine on the processes leading to morphine-induced reward-seeking behavior in Sprague-Dawley rats. Methods: The model of CPP was used to assess the rewarding effect of morphine The levels of histamine, glutamate, γ-aminobutyric acid (GABA), dopamine (DA) and 3,4-dihydroxyphenyl-acetic acid (DOPAC) in rat brains were measured with high-performance liquid chromatography. Immunohistochemistry technique was used to observe themorphological changes of neurons. Results: Intraperitoneal injection of mor-phine (2,5 or 10 mg / kg) induced the development of CPP in a dose- dependent manner. In addition, morphine administrations (10 mg / kg) decreased the hista-mine content and reduced the number and size of histaminergic neurons in the tuberomammillary nucleus (TM), as well as markedly increasing the DOPAC / DAratios in the ventral tegmental area (VTA) and nucleus accumbens (NAc). Intra-peritoneal injection of histidine r 200 mg / kg) dose-dependently inhibited the development of morphine-induced CPP.Bilateral lesions of the TM, which created the histamine levels in the VTA and NAc, potentiated the development of CPP induced by morphine (1 mg / kg, a dose that produced no appreciable effectwhen given alone) and increased the DOPAC / DA ratios in the VTA and NAc, but do not change the glutamate or GABA levels in these nuclei. Histidine reversed the effects of the TM lesions. Confc: These results indicate that endog-enous histamine plays a role in inhibiting the development of morphine-induced reward-seeking behavior, and the inhibition may involve the modulation of dopa-minergic activity.
其他文献
在儿科治疗中,静脉滴注葡萄糖广为应用,尤其在儿童消化不良或新生儿脱水热时,为纠正脱水及给予抗生素而输入葡萄糖。但平时一般很少注意由此而引起的血糖水平失衡,尤其是低
本文应用质量动替代法,采用质量分布和附加齿轮机构与凸轮弹簧机构,以stephenson型六杆机构为例对平面多杆机构的摆动力、摆动力矩和输入扭矩进行了完全平衡。 In this pape
目的:探讨Th1/Th2淋巴细胞偏移对大鼠睾丸缺血再灌注损伤的影响。方法:SD雄性大鼠30只,随机分成假手术组、睾丸扭转组、扭转复位组,每组10只,通过建立左侧睾丸扭转和复位动物
Aim:To determine whether the anti-inflammatory effect of minocycline on postis-chemic brain injury is mediated by the inhibition of 5-lipoxygenase (5-LOX)expre
本文通过不同分子量的高分子量聚合物(部分水解聚丙烯酰胺)在不同渗透率岩心中的流动实验,研究了高分子量聚合物的分子量与岩心渗透率之间的匹配关系,为大庆油田采用高分子量聚合
液氮助排技术,是采用延迟胶联技术在压裂液的前置液中加入氮气,形成均匀泡沫冻胶,用来撑开地层,并且在压裂后,靠释放出的氮气反推破胶水化液排出地层,提高压裂液的返排率,减
我厂煤场仅有一台哈尔滨重型机器厂生产的DQ3025堆取料机,自1982年安装运行以来,由于存取煤任务重,悬臂在各个方位工作时间不均匀,使回转机构的交叉滚子轴承严重磨损且磨损
在中小学教育中,学生是学习活动不可替代的主体。学生主动性发展的最高水平是能动、自觉地规划自身的发展,成为自己发展的主人,这是教育成功的重要标志。教师应承认每一个学生都具有自己的独特性,一个真正出色的教师,应该以学生发展为本,视学生为独立的个体,研究学生的需要、兴趣、性向。在教学中,教师应该通过自己创造性的教学,努力促进学生素质的提高,使学生真正成为德、智、体、美全面发展的一代新人。教师应当以学生发
大气、霸道、沉稳、成熟、领袖气质……提到这些词语你会想到什么?不不,不是奥巴马,我们今天文章的主角当然是汽车。想到了吧,没错,能配得上这些溢美之词的只能有一个品牌—
科技奖励是国家科技政策的重要组成部分,对国家科学技术的发展起着举足轻重的作用,受到世界各国的高度重视和普遍关注.自建国以来,我国就十分重视科技奖励工作及其研究,经过