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本文报告了硝基乙烯基吲哚类化合物抗溶组织内阿米巴的作用。作者采用Dutta和Yadava改良法将TP S-I Diamond培养基中生长的NIH:200株无菌溶组织内阿米巴进行体外试验,观察3-(2-硝基乙烯基)吲哚、1-甲基-3-(2-硝基乙烯基)吲哚、3-(2-甲基-2-硝基乙烯基)吲哚、1-甲基-3-(2-甲基-2-硝基乙烯基)吲哚、3-甲酰吲哚、1-甲基3-甲酰吲哚及5-硝基-3-甲酰吲哚等化合物的体外抗阿米巴作用。与甲硝唑作比较,结果显示3-(2-硝基乙烯基)吲哚具有很强的抗阿米巴活性,其最小抑制浓度
This article reports the role of the nitrilotriacetamides against Entamoeba histolytica. The authors used Dutta and Yadava modified method to in vitro test NIH: 200 strains of Entamoeba histolytica grown in TP SI Diamond medium to observe 3- (2-nitrovinyl) indole, 1-methyl 3- (2-nitrovinyl) indole, 3- (2-methyl-2-nitrovinyl) Yl) indole, 3-formylindole, 1-methyl 3-formylindole and 5-nitro-3-formylindole in vitro. Compared with metronidazole, the results showed that 3- (2-nitrovinyl) indole has a strong anti-amoebic activity, the minimum inhibitory concentration