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pinacidil(吡那地尔)是胍/硫脲类钾通道开放剂,为消旋体。Lemakalim(BRL38227)为苯并吡喃类钾通道开放剂,为Cromakalim的左旋体。国外近几年已开展了关于这类药物的研究,主要探讨其在治疗心血管疾病等方面的药理作用。但国内对此研究报道还较少,尤其对Lemakalim。本实验通过观察Pinacidil和Lemakalim
Pinacidil (pinacidil) is a guanidine / thiourea potassium channel opener, racemate. Lemakalim (BRL38227) is a benzopyran-like potassium channel opener, the L-form of Cromakalim. In recent years, foreign countries have carried out research on such drugs and mainly discussed their pharmacological effects in the treatment of cardiovascular diseases. However, there are few reports about this in China, especially for Lemakalim. This experiment by observing Pinacidil and Lemakalim