螠蛏共附枯草芽孢杆菌110次级代谢产物的抑菌抗肿瘤活性研究

来源 :中国海洋药物 | 被引量 : 0次 | 上传用户:qqllql
下载到本地 , 更方便阅读
声明 : 本文档内容版权归属内容提供方 , 如果您对本文有版权争议 , 可与客服联系进行内容授权或下架
论文部分内容阅读
目的检测螠蛏共附枯草芽孢杆菌110次级代谢产物的抑菌活性组分,并探讨抑菌活性组分的抗肿瘤作用。方法用0.22μm滤膜过滤将螠蛏共附枯草芽孢杆菌110的菌体和发酵液分开,用硫酸铵沉淀发酵液的蛋白组分并用SDS-PAGE检测,用滤纸片法分别检测菌株发酵液、菌体及胞外蛋白的抑菌活性,琼脂块法检测抑菌活性组分的抑真菌活性,用海虾毒性法和MTT法检测抑菌活性组分的抗肿瘤活性。结果螠蛏共附枯草芽孢杆菌110的发酵液抑菌活性远远高于菌体的抑菌活性,发酵液的硫酸铵沉淀物具有很强的抑菌活性,硫酸铵沉淀的110活性粗蛋白主要由分子量约为60、45和25kDa的3条带组成。110活性粗蛋白对8种真菌指示菌具有抑制作用,其中对辣椒青枯、番茄灰霉和瓜类枯萎的抑菌圈直径超过20mm。该活性粗蛋白还对白血病细胞K562、肝癌细胞HepG-2和人乳腺癌细胞MDA-MB-231具有抑制作用,其中200μg/mL的蛋白对人肝癌细胞HepG-2抑制率达74.01%。结论螠蛏共附枯草芽孢杆菌110胞外蛋白有抗肿瘤活性和广谱抑菌活性,具有潜在的开发价值。 Objective To detect the antibacterial activity components of secondary metabolites of Bacillus subtilis 110 and to study the anti-tumor effect of antibacterial activity components. Methods The bacterial cells and fermentation broth of Bacillus subtilis 110 were separated by filtration with 0.22 μm membrane filter. The protein components of the fermentation broth were precipitated by ammonium sulfate and detected by SDS-PAGE. The fermentation broth of the strains was detected by filter paper method. The antibacterial activity of the bacterium and the extracellular protein was tested. The fungistatic activity of the antibacterial activity component was detected by the agar block method. The antitumor activity of the antibacterial activity component was tested by shrimp toxicity method and MTT method. Results The antibacterial activity of the fermentation broth of Bacillus subtilis 110 was much higher than that of the bacterium. The ammonium sulfate precipitate of the fermentation broth had strong antibacterial activity. The crude protein precipitated by ammonium sulfate was mainly Consists of three bands with molecular weights of about 60, 45 and 25 kDa. 110 active crude protein had inhibitory effect on eight fungi. Among them, the inhibition zones of withered pepper, tomato gray mold and melon were more than 20mm in diameter. The active crude protein also has inhibitory effects on K562 leukemia cells, HepG-2 hepatoma cells and MDA-MB-231 human breast cancer cells. The inhibitory rate of 200μg / mL protein on HepG-2 cells was 74.01%. Conclusion The total protein of Bacillus subtilis 110 extracellular protein has anti-tumor activity and broad-spectrum antibacterial activity, which has potential value for development.
其他文献
目的在生物活性和化学方法指导下,从1株海兔来源真菌Aspergillus terreus(RA29-5)中分离鉴定海洋天然产物,并对其进行生物活性评价。方法运用硅胶柱层析、Sephadex LH-20凝胶
芋螺毒素由芋螺毒液管和毒囊内壁的毒腺所分泌,每种芋螺的毒液中至少含50~200种活性多肽。根据芋螺毒素高度保守的信号肽序列及二硫键骨架,芋螺毒素分为A、B1、B2、B3、C、D
真菌产生的次级代谢产物是新药开发的重要资源,其生物合成过程受到众多因素的调控.化学表观遗传操作是利用小分子化学物质抑制真菌中影响表现遗传的酶类,激活沉默的生物合成
  本文研究了这两种技术在数字博物馆的应用,分析其核心的应用技术.这些技术的应用必将推动数字博物馆的建设达到新的水平。
  本文应用目前的IBM技术对良渚文物进行基于照片三维重构,通过使用定标板,较好的解决了照相机的定标问题,取得了较好的定标精度,本文还详细讨论了实验过程中所采
会议
目的观察海兔素(Aplysin)对酒精性肝损伤大鼠肝组织Fas、FasL表达及血清肿瘤坏死因子-α(TNF-α)水平的影响。方法50只雄性Wistar大鼠随机分为5组。正常对照组,每日灌胃生理
目的研究海洋小球藻多糖的制备工艺及其抑制肿瘤血管生成的作用。方法比较多种提取方法提取多糖,确定最适提取工艺,经乙醇沉淀,并结合DEAE-Cellulose 52柱色谱分离纯化;采用
  本论文讨论了我国文化遗产的现状,基于图像绘制技术(IBR)和地理信息系统(GIS)的方法与特点,提出了一种基于图像绘制与GIS集成系统,以及该系统在文化遗产旅游和保护领域中
本文从自动测试系统的发展过程,分析了第三代自动测试系统的结构模式,提出了建立在IBM-PC总线基础上的新型实用结构模式,且利用这种模式,组建并实现了鱼雷自动测试系统。 Ba
先进的采用y-系数法的噪声系数测量仪可同时测量增益和噪声系数,并可以自动修正第二级的影响。这要求二端口的输出端要匹配。非匹配的器件需要一个输出调配器。本文介绍了一