All-trans retinoic acid inhibited angiotensin Ⅱ-induced increase in cell growth and collagen secreti

来源 :Acta Pharmacologica Sinica | 被引量 : 0次 | 上传用户:woaiwojiaren5210
下载到本地 , 更方便阅读
声明 : 本文档内容版权归属内容提供方 , 如果您对本文有版权争议 , 可与客服联系进行内容授权或下架
论文部分内容阅读
Aim:To determine whether all-trans retinoic acid(atRA)acts to modulate angio-tensin Ⅱ(Ang Ⅱ)-induced cardiac fibroblast cell growth and collagen secretion.Methods:Cultured neonatal rat cardiac fibroblasts(CF)were used in the experiment.A 3-(4,5-dimethylthiazol-2-yl)-2,5-diphenyl tetrazolium bromide(MTT)assay wasused to detect cell growth of the CF;and immunocytochemistry and Westernblotting were used to measure the production and secretion of collagen and theexpression of transforming growth factor-β_1(TGF-β_1)by the CF.Results:atRA(1×10~(-7) to 1×10~(-5) mol/L)inhibited the Ang Ⅱ-induced increase in cell growth of CF(P<0.05).Ang Ⅱ stimulated the secretion of collagen types Ⅰ and Ⅲ by the CF.This effect was blocked by AT_1 receptor antagonist losartan(1×10~(-6) mol/L),butnot by AT_2 receptor antagonist PD 123319 (up to 1×10~(-6) mol/L).Exposure of CF toatRA(1×10~(-5) mol/L)attenuated the Ang Ⅱ-induced increase in the secretion ofcollagen types Ⅰ and Ⅲ(P<0.05).atRA (1×10~(-5) mol/L)also blocked the Ang Ⅱ-induced increase in the expression of TGF-β_1.Conclusion:atRA inhibits the AngⅡ-induced increase in cell growth and collagen secretion of neonatal rat CF.Theeffect of atRA is possibly mediated by lowering the TGF-β_1 level.These observa-tions support the notion that atRA is a potential candidate for the prevention andtherapy of cardiac remodeling. Aim: To determine whether all-trans retinoic acid (atRA) acts to modulate angio-tensin II (Ang II) -induced cardiac fibroblast cell growth and collagen secretion. Methods: Cultured neonatal rat cardiac fibroblasts (CF) were used in the experiment. A 3- (4,5-dimethylthiazol-2-yl) -2,5-diphenyl tetrazolium bromide (MTT) assay was used to detect cell growth of the CF; and immunocytochemistry and Western blotting were used to measure the production and secretion of collagen and theexpression of transforming growth factor-β_1 (TGF-β_1) by the CF. Results: atRA (1 × 10 -7 to 1 × 10 -5 mol / L) inhibited the Ang Ⅱ-induced increase in cell growth of CF (P <0.05). Ang Ⅱ stimulated the secretion of collagen types Ⅰ and Ⅲ by the CF.This effect was blocked by AT_1 receptor antagonist losartan (1 × 10 -6 mol / L), butnot by AT_2 receptor antagonist PD 123319 (up to 1 × 10 -6 mol / L) .Exposure of CF toatRA (1 × 10 -5 mol / L) attenuated the Ang Ⅱ-induced increase in the secretion ofcollagen types Ⅰ and Ⅲ (P <0.05) .a tRA (1 × 10 ~ (-5) mol / L) also blocked the Ang Ⅱ-induced increase in the expression of TGF-β_1.Conclusion: atRA inhibits the AngⅡ-induced increase in cell growth and collagen secretion of neonatal rat CF. Theeffect of atRA is possibly mediated by lowering the TGF-β_1 level. The observa-tions support the not that that atRA is a potential candidate for the prevention and treatment of cardiac remodeling.
其他文献
5月的古城丹阳,洋溢着浓浓春意。在丹凤影剧院召开的为市民广场建设捐资大会上,一位中等身材,双目炯炯有神,充满睿智与精明的企业家,高高地举起了捐资10万元的标牌,会场上顿
顺向断鼻是断陷盆地一种普遍的构造类型,但顺向断鼻有时成藏,有时不成藏,其成藏条件颇有争论,并直接影响其评价和钻探。以冀中坳陷南部的束鹿凹陷为例,参考其它地区,归纳了影
本文用金属材料预钝化处理、金属表面涂覆层、添加缓蚀剂及阳极保护方法,控制钛在硫酸铝溶液中的腐蚀。试验结果表明,上述4种方法对钛在该体系中腐蚀都有一定控制作用,以阳极
在独山脚下,白河之滨,南阳的东大门,人们以惊异的目光注视着这里的变化,这就是南阳交通驾校——经省交通厅批准的全市惟一一家事业性培训机动车驾驶员的专业学校。她以娇美
Aim:To investigate whether tanshinone ⅡA could improve the effect of UWsolution for skeletal muscle preservation and to determine the dose range oftanshinone
钎焊是铝合金重要的联接工艺,但与其它金属相比,铝合金钎焊有一定的难点。现探索出一种简便、廉价铝合金钎焊工艺,钎焊质量优良,介绍如下:1.采用锌钎料。如没有现成的锌钎料,可用一般
Aim:To elucidate the molecular nature of sulfhydryl modification by hydrogenperoxide on type 1 ryanodine receptor(RyR1).Methods:Rabbit skeletal musclesarcoplas
直线度公差是控制机械零件平面形状的一项重要技术指标。零件平面的精度不论高低,它的实际误差是必须测定的。只有知道了误差,才能判断其是否合格,才能进一步分析产生误差的
深圳求实技术开发有限公司总经理张凤球女士于1985年发明了一种新型的储油罐内浮顶——“张氏浮盘”,该项技术已先后获得中国和美国专利,美国石油界命名其为“张氏浮盘”。
安痛定为解热镇痛药,具有退热、镇痛作用,在临床上广泛使用。我院遇一例患者因使用安痛定引起过敏性休克,现报告如下: 病例:患儿,女性,5岁。主因感冒于92年3月7日来我院门诊