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目前最有效的抗雄激素药为醋酸赛普龙(Cyprote rone acetate,CPA),另外,赛普龙(Cyproterone,CP)和非甾体制剂氟化酰胺(Flutamide)也具有抗雄激素作用(见图1)。
Cyproterone (CP) and Flutamide, the non-steroidal anti-androgen agent, also have anti-androgenic effects figure 1).