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盐酸二氢埃托菲是我国研究成功的高效镇痛药物,它是迄今为止作用最强的镇痛剂,其镇痛活性是吗啡的1000倍。盐酸二氢埃托菲舌下含服5分种后见效,镇痛作用持续4~6小时。主要用于各种原因引起的疼痛,尤其是晚期癌症的止痛,其止痛率可达90%。盐酸二氢埃托菲还可用于海洛因等毒品的戒毒,其机制是因为盐酸二氢埃托菲是阿片受体的强激动剂,而阿片受体分几个不同类型,研究揭示:盐酸二氢埃托菲作用的阿片受体可能不是介导成瘾的
Dihydroetofenhydrochloride is a highly effective analgesic which has been successfully researched in China. It is by far the most effective analgesic and its analgesic activity is 1000 times that of morphine. Hydrochloride emodin sublingual sublingual 5 minutes after the effective, analgesic effect lasted 4 to 6 hours. Mainly used for various causes of pain, especially in advanced cancer pain, the pain rate up to 90%. Dihydroteethane dihydrochloride can also be used for drugs such as heroin detoxification, the mechanism is because dihydroetorphine dihydrochloride is a strong agonist of opioid receptors, and opioid receptors divided into several different types, the study revealed: dihydrogen hydrochloride Opioid receptors that actofetofen may not mediate addiction