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研究了扑热息痛微型灌肠剂与口服片剂、肌肉注射剂在家兔上的相对生物利用度。认为微型灌肠剂生物利用度优于口服片剂,是扑热息痛一种合适剂型。
The relative bioavailability of paracetamol mini enema to oral tablets and intramuscular in rabbits was studied. The mini-enema bioavailability is considered superior to oral tablets and is a suitable dosage form for paracetamol.