比较蛋白质组学分析揭示消癌解毒方含药血清作用人肝癌SMMC-7721细胞差异蛋白表达

来源 :中华中医药杂志 | 被引量 : 0次 | 上传用户:kuangyunlo
下载到本地 , 更方便阅读
声明 : 本文档内容版权归属内容提供方 , 如果您对本文有版权争议 , 可与客服联系进行内容授权或下架
论文部分内容阅读
目的:观察消癌解毒方含药血清对人肝癌细胞SMMC-7721细胞中蛋白表达变化的影响。方法:选择人肝癌SMMC-7721细胞作为实验对象,消癌解毒方含药血清作用人肝癌SMMC-7721细胞24h后,采用TMT肽段标记,质谱鉴定分析,运用IPA软件对结果进行生物信息学分析,观察用药前后各组蛋白质表达的差异,应用Western blot法检测Cytochrome C、Caspase-3、Cleaved-Caspase-3蛋白的表达。结果:共鉴定出3 025个蛋白点,消癌解毒方各剂量组与模型组相比差异表达明显的蛋白423个,其中消癌解毒方高剂量组负调控蛋白55个,正调控蛋白85个;消癌解毒方中剂量组负调控蛋白33个,正调控蛋白50个;消癌解毒方低剂量组负调控蛋白36个,正调控蛋白49个;顺铂组负调控蛋白38个,正调控蛋白77个。这些差异表达蛋白涉及脂质代谢、凋亡、氧化应激等方面。信号通路分析涉及Granzyme A Signaling、TR/RXR Activation等通路。Western blot结果显示消癌解毒方处理人肝癌SMMC-7721细胞24h后可引起Cytochrome C蛋白被释放,Cleaved-Caspase-3蛋白表达量上调,Caspase-3蛋白表达量下调。结论:消癌解毒方作用于人肝癌SMMC-7721细胞有多靶点,多中心的调控作用,其中激活线粒体凋亡相关蛋白可能是其抑制肿瘤生长,诱导肿瘤凋亡的途径之一。 Objective: To observe the effect of Xiaoyan Jiedu Fang containing serum on the protein expression of human hepatoma SMMC-7721 cells. Methods: Human hepatocellular carcinoma SMMC-7721 cells were selected as experimental subjects. Human hepatocellular carcinoma SMMC-7721 cells were treated with Xiaojian Jiedu decoction for 24 h. The results were analyzed by mass spectrometry (TMT) and identified by bioinformatics analysis using IPA software The difference of protein expression in each group before and after treatment was observed. Western blot was used to detect the expression of Cytochrome C, Caspase-3 and Cleaved-Caspase-3. Results: A total of 3 025 protein spots were identified. There were 423 differentially expressed proteins in each dose group of Xiaoyao Jiedu Fang compared with the model group. Among them, there were 55 negative regulators and 55 positive regulators The negative control protein of Xiaowangjiedu Fang middle dose group had 33 negative regulators and 50 positive regulators, while the negative control Xiaowangjiedu Fang low dose of 36 negative regulators, positive regulators of 49 and negative regulators of cisplatin 38 positive regulators 77 proteins. These differentially expressed proteins involved in lipid metabolism, apoptosis, oxidative stress and so on. Pathway analysis involves access to Granzyme A Signaling, TR / RXR Activation and more. Western blot results showed that Cytochrome C protein was released by Xiaojian Jiedu Fang treatment of human hepatocellular carcinoma SMMC-7721 cells for 24h, the expression of Cleaved-Caspase-3 protein was up-regulated and the expression of Caspase-3 protein was down-regulated. Conclusion: Xiaojian Jiedu Fang can inhibit the proliferation of human hepatocellular carcinoma SMMC-7721 cells and induce the apoptosis of SMMC-7721 cells. The activation of mitochondrial apoptosis-related proteins may be one of the pathways of inhibiting tumor growth and inducing tumor apoptosis.
其他文献
目的:观察新风胶囊对佐剂型关节炎(AA)大鼠肺功能、肺组织氧化应激状态及Keap1-Nrf2/ARE信号通路表达的影响. 方法:48只雄性SD大鼠按随机数字表随机分为正常组(NC),模型组
会议
乏燃料组件池边检査是核电站燃料组件必不可少的重要检测项目.针对国内外池边检查技术发展现状的不足,设计了一套基于摄影测量的乏燃料组件池边检查系统,结合接触式与非接触
慢性扁桃腺肿大是上呼吸道系统的多发病,在临床上发病率日渐增高,其中滥用、过用抗生素及大量清热解毒药是常见诱因,严重影响患者的生活质量.从中医角度探讨抗生素及清开灵等
"精准医疗"是时下国内最受关注和热议的话题.文章参考"精准医疗"新模式,以大数据采集、大数据处理、准确化诊断与个性化治疗为结合点,发挥中医自古以来辨证论治和个性化诊疗
目的:体外研究双氢青蒿素(DHA)对人肝星状细胞(HSCs)坏死性凋亡的影响及机制. 方法:HSCs分为对照组以及DHA处理组.应用噻唑蓝(MTT)、细胞计数试剂盒-8(CCK-8)以及亚甲基蓝
会议
五脏是机体应时而变并在所应季节起主要调节作用的时间调节系统。脏腑在当旺的季节,其生理功能随着所应季节的阴阳消长出现增强或减弱,并对其他脏腑处于支配地位,发挥着对脏
作为一种新型焊接方法,局部真空电子束焊接常被用于制造厚大的奥氏体不锈钢焊接接头,而该类接头的焊接残余应力和变形问题受到广泛关注.对板厚40 mm的SUS310S不锈钢局部真空
机床误差是导致圆弧齿线圆柱齿轮齿面误差的主要原因,研究机床误差与齿面误差之间的关系将为机床加工参数反求、齿面误差修正等提供理论依据.基于圆弧齿线圆柱齿轮成型原理建
空间意识的形成需要长期的努力和教学环节的保证,是一个学生一开始绘画训练就应该接触到的问题。从我国绘画教学的总体情况上看,对造型的探讨基本上是在焦点透视的空间框架下展
提出一种用于精密线性位移台滚转角和运动直线度同步测量的激光外差干涉系统.该干涉系统由一个Koster棱镜、角隅棱镜、分光镜、1/2波片、直角棱镜、1/4波片以及楔面棱镜和楔