Chemical Mutations on Specific Nucleobases as a Feasible Approach for More Efficient DNAzymes

来源 :第九届IUPAC化学生物学国际研讨会暨第八届世界华人药物化学研讨会 | 被引量 : 0次 | 上传用户:pgwork2011
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  Residue replacement of functional nucleic acids is the first choice for their structure-activity relationship and better performance,in the absence of active conformation.Two small DNAzymes,10-23 as genetic therapeutics against many disease-related genes and 8-17 DNAzyme as biosensors,have been studied extensively.Canonical residue replacement and deletion confirmed the conservation of the catalytic cores,and no better analogs could be obtained by this way.
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