2-Pyridone Based Antimalarials Synthesis and Activity

来源 :IUPAC 9th International Conference on Novel Materials and th | 被引量 : 0次 | 上传用户：ccwawa

【摘要】

：

A new class of compounds with the envisaged ability to inhibit cysteine proteases,especially of Plasmodium, [1] was designed, based on a 2-pyridone scaffold.Ami

【作者】

：

T.van Ree S.A.Nethavhani

【机构】

：

SchoolofMathematicalandNaturalSciences,UniversityofVenda,Thohoyandou0950,SouthAfrica

【出处】

：

IUPAC 9th International Conference on Novel Materials and th

【发表日期】

：

2013年10期

【关键词】

：

Dipeptide mimic malaria 2-pyridone

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A new class of compounds with the envisaged ability to inhibit cysteine proteases,especially of Plasmodium, [1] was designed, based on a 2-pyridone scaffold.Amino acid residues such as phenylalanine and valine were included [2].

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2-Pyridone Based Antimalarials Synthesis and Activity

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