One-pot synthesis of 4-methylisoquinolines via sequential Pd-catalyzed Heck reaction and intramolecu

来源 :全国药物化学学术会议暨第四届中英药物化学学术会议 | 被引量 : 0次 | 上传用户：zhangsonghuan

【摘要】

：

An efficient,one-pot synthesis of 4-methylisoquinolines via a cascade Pd-catalyzed Heck reaction,intramolecular cyclization and isomerization has been developed.

【作者】

：

Yulin Tian Jianguo Qi Chenbin Sun Dali Yin Xiaojian Wang Qiong Xiao

【机构】

：

State Key Laboratory of Bioactive Substances and Functions of Natural Medicines,Institute of Materia

【出处】

：

全国药物化学学术会议暨第四届中英药物化学学术会议

【发表日期】

：

2013年11期

【关键词】

：

One-pot 4-Methylisoquinoline Heck reaction

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　　An efficient,one-pot synthesis of 4-methylisoquinolines via a cascade Pd-catalyzed Heck reaction,intramolecular cyclization and isomerization has been developed.

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One-pot synthesis of 4-methylisoquinolines via sequential Pd-catalyzed Heck reaction and intramolecu

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