The Synthesis of Ipriflavone Analogues as Anti-osteoclastogenesis Agents

来源 :第九届IUPAC化学生物学国际研讨会暨第八届世界华人药物化学研讨会 | 被引量 : 0次 | 上传用户:nike880713
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  The inflammatory cytokines play a major role in osteoclastogenesis and lead to the bone resorption that is frequently associated with osteoporosis.Ipriflavone has been reported possessed anti-inflammatory activity.The ipriflavone analogues were synthesized and investigated the anti-osteoclastogenesis activity.The series of compounds was subjected to inhibit nuclear factor kappa B ligand (RANKL) plus macrophage colony stimulating factor0induced osteoclatic differentiation from bone marrow stromal cells and RAW264.7 macrophage cells.The ipriflavone analogues,7-fluoroisoflavnoes,were shown benefited bone health by attenuating bone loss through inhibiting the osteoclast.
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