Simotinib as modulator of P-glycoprotein: substrate, inhibitor or inducer?

来源 :2015年中国药物制剂大会、中国药学会药剂专业委员会2015年学术年会暨国际控释协会中国分会2015年学术年会 | 被引量 : 0次 | 上传用户：m2564

【摘要】

：

　　Purpose: Effiux transporters play a significant role in chemotherapy drug resistance.Interaction between these transporters, such as P-glycoprotein (P-gp),

【作者】

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Lingling Huang Pei Li Cheng Shen Zeneng Cheng Qubo Zhu

【机构】

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The School of Pharmaceutical Sciences in Central South University

【出处】

：

2015年中国药物制剂大会、中国药学会药剂专业委员会2015年学术年会暨国际控释协会中国分会2015年学术年会

【发表日期】

：

2015年期

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　　Purpose: Effiux transporters play a significant role in chemotherapy drug resistance.Interaction between these transporters, such as P-glycoprotein (P-gp), and drugs might influence their pharmacological properties and toxicities.

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Simotinib as modulator of P-glycoprotein: substrate, inhibitor or inducer?

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