SM02-P22:Discovery of novel Kv1.5 potassium channel blockers using structure-based drug design strat

来源 :第13届亚洲化学大会(13th Asian Chemical Congress) | 被引量 : 0次 | 上传用户:easelin
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  During recent years, Atrial Fibrillation (AF) is emerging as a major public health problem among the aging population.The ultra-rapid delayed rectifier potassium current (IKur), encoded by Kv 1.5 gene, is a selective target for the treatment of AF.Therefore, several pharmaceutical companies have made their efforts in developing selective Kvl.5 blockers by taking some deeper insight into action mechanism and structural information.
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